Skip to main navigation Skip to search Skip to main content

Synthesis of 4-oxo and 4-hydroxyimino-4-deoxy-Kdn2en derivatives

  • Xue Sun
  • , Toshitsugu Kai
  • , Noriko Sato
  • , Hiroaki Takayanagi
  • , Kimio Furuhata
  • Kitasato University

Research output: Contribution to journalArticlepeer-review

1 Scopus citations

Abstract

2,6-Anhydro-3-deoxy-D-manno-non-2-en-4-ulosonic acid (4-oxo-Kdn2en, 2) was synthesized from methyl 2,6-anhydro-3-deoxy-D-glycero-D-galacto-non-2-enonate (Kdn-2en methyl ester, 7) by the oxidation with manganese dioxide in dry acetone in good yield. 4-Hydroxyimino-Kdn2en derivatives (3), and 4-carbethoxymethylene-Kdn2en derivatives (4) were synthesized from the peracetylated methyl ester of 4-oxo-Kdn2en by oximation and Wittig reaction in good yield, respectively.
Original languageEnglish
Pages (from-to)1131-1138
Number of pages8
JournalJournal of Carbohydrate Chemistry
Volume18
Issue number9
DOIs
StatePublished - Jan 1 1999

Cite this